Zidovudine (retrovir)-
â—‹ Non-nucleoside reverse transcriptase inhibitor
â– Only one can be given IV intrapartum (need for this based on viral
load) → considered drug of choice in pregnancy
â—‹ Penetrates CSF
â—‹ Adverse effects:
â– Hematologic toxicity
â— Hold for Hgb below 5 gm/dL or 25% drop from baseline
â— Hold for neutrophil count below 750 cells/mL